Sulfonylalkanoylamino hydroxyethylamino sulfonamide...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

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Details

C514S367000, C514S375000, C514S464000, C514S469000, C544S135000, C544S137000, C546S196000, C546S198000, C548S178000, C548S217000, C548S517000, C548S518000, C549S434000, C549S438000, C549S467000

Reexamination Certificate

active

07045518

ABSTRACT:
Selected sulfonylalkanoylamino hydroxyethylamine sulfonamide compounds are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease. The present invention relates to such retroviral protease inhibitors and, more particularly, relates to selected novel compounds, composition and method for inhibiting retroviral proteases, such as human immunodeficiency virus (HIV) protease, prophylactically preventing retroviral infection or the spread of a retrovirus, and treatment of a retroviral infection.

REFERENCES:
patent: 4450164 (1984-05-01), Bristol et al.
patent: 4477441 (1984-10-01), Boger et al.
patent: 4514391 (1985-04-01), Gordon et al.
patent: 4548926 (1985-10-01), Matsueda et al.
patent: 4595407 (1986-06-01), Carter
patent: 4599198 (1986-07-01), Hoover
patent: 4616088 (1986-10-01), Ryono et al.
patent: 4634465 (1987-01-01), Ehrenfreund et al.
patent: 4668769 (1987-05-01), Hoover
patent: 4668770 (1987-05-01), Boger et al.
patent: 4757050 (1988-07-01), Natarajan et al.
patent: 4880938 (1989-11-01), Freidinger
patent: H725 (1990-01-01), Gordon
patent: 4963530 (1990-10-01), Hemmi et al.
patent: 4977277 (1990-12-01), Rosenberg et al.
patent: 5705500 (1998-01-01), Getman et al.
patent: 5985870 (1999-11-01), Getman et al.
patent: 6169085 (2001-01-01), Getman et al.
patent: 6380188 (2002-04-01), Getman et al.
patent: 6667307 (2003-12-01), Getman et al.
patent: 0 104 041 (1984-03-01), None
patent: 0 114 993 (1984-08-01), None
patent: 0 172 347 (1986-02-01), None
patent: 0 223 437 (1987-05-01), None
patent: 0 264 795 (1988-04-01), None
patent: 0 342 541 (1989-05-01), None
patent: 0 337 714 (1989-10-01), None
patent: 0 346 847 (1989-12-01), None
patent: 0 356 223 (1990-02-01), None
patent: 0 389 898 (1990-10-01), None
patent: 0 393 445 (1990-10-01), None
patent: 0 393 457 (1990-10-01), None
patent: 0 402 646 (1990-12-01), None
patent: 0 468 641 (1992-01-01), None
patent: 2184730 (1987-07-01), None
patent: 2200115 (1988-07-01), None
patent: 2209752 (1989-05-01), None
patent: 84/03044 (1984-08-01), None
patent: WO 92/00750 (1992-01-01), None
patent: 92/08699 (1992-05-01), None
patent: 93/13066 (1993-07-01), None
patent: 94/04493 (1994-03-01), None
patent: 94/08458 (1994-05-01), None
patent: 94/10136 (1994-05-01), None
patent: WO 95 06030 (1995-03-01), None
patent: WO 95 33464 (1995-12-01), None
International Search Report of PCT/US96/02682 dated Aug. 21, 1996.
Roberts et al.,Science, 248, 358 (1990).
Erickson et al.,Science, 249, 527 (1990).
Pearl et al.,Nature328 (1987).
Martin, Drugs of the Future, (1991), 16(3), 210-212.
Meek et al.,Nature, 343:90-92, (1990).
McQuade et al.,Science, 274, 454 (1990).
Rich et al., Pept. Struct. Funct. Am. Pept. Sym. 8th ed. pp. 511-520 (1983).
Rosenberg et al.,J. Med. Chem., 30, 1224-1228 (1987).
Fittkau,J. Prakt. Chem. 315, 1037 (1973).
Hirsh et al.,N. Eng. J. Med., 328, 1686 (1993).
E. E. Gilbert, “Recent Developments in Preparative Sulfonation and Sulfation,”Synthesis, 3 (1969).
Mitsuya et al.,Proc. Natl. Acad. Sci. USA, 83, 1911-15 (1986).
Silcox et al.,J. Heterocycl Chem., 4, 166-67 (1967).
Cabiddu et al.,Synthesis, 797-798 (1976).
Ncube et al.,Tet. Lett, 26, 2345-2348 (1978).
Ncube et al.,Tet. Lett, 3, 255-256 (1977).
Cole et al.,Aust. J. Chem., 33, 675-80 (1980).

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