Cyclopentenedione antifungal compounds and methods for their...

Organic compounds -- part of the class 532-570 series – Organic compounds – Oxygen containing

Reexamination Certificate

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

C514S684000, C514S687000

Reexamination Certificate

active

07109380

ABSTRACT:
Compounds and methods useful in the control, treatment, and prevention of fungal activity, of the following formula:where R1-3are independently H, alkyl, methyl, acyl, halogen, phenyl, R4is H, alkyl, methyl, acyl, alkoxy, halogen, phenyl provided that when R3is methyl and R4is H, R1and R2are not both H; and stereoisomers, analogs, and pharmaceutically acceptable salts thereof.

REFERENCES:
patent: 3852470 (1974-12-01), Grohe et al.
patent: 6844353 (2005-01-01), Wedge et al.
patent: 2140737 (1973-02-01), None
patent: 2248819 (1974-04-01), None
patent: 2804271 (1998-08-01), None
patent: 51019125 (1976-02-01), None
patent: 52079022 (1977-07-01), None
patent: 53101336 (1978-09-01), None
patent: WO99/04777 (1999-02-01), None
Kiang, H. H.; Sim, K. Y. J. Chem. Soc. 1962, 4338.
Lee, H. H. Tetrahedron Lett. 1968, 4243.
Liu, S. Y.; Ogihara, Y. Yakugaku Zasshi 1975, 95, 114.
Leong, et al., J. D. Phytochemistry 1998, 47, 891.
Aoyama, et al.; Bioorg. Med. Chem. Lett. 2001, 11, 1695.
Inayama, S.; Mamoto, K.; Shibata, T.; Hirose, T. J. Med. Chem. 1976, 19, 433.
Shestak, P.; Novikov, V. L.; Stekhova, S. I.; Gorshkova, I. A. Pharm. Chem. J. 1999, 33, 18.
Hori, H.; Nagasawa, H.; Ishibashi, M.; Uto, Y.; Hirata, A.; Saijo, K.; Ohkura, K.; Kirk, K. L.; Uehara, Y. Bioorg. Med. Chem. 2002, 10, 3257.
Watanabe, M.; Hisamatsu, S.; Hotokezaka, H.; Furukawa, S. Chem. Pharm. Bull. 1986, 34, 2810.
Kalinin, A. V.; Snieckus, V. Tetrahedron Lett. 1998, 39, 4999.
Bruce, J. M.; Creed, D.; Dawes, K. J. Chem .Soc. (C) 1971, 3749.
Irngartinger, H.; Stadler, B. Eur. J. Org. Chem. 1998, 605.
Brehm, I.; Meier, H. Eur. J. Org. Chem. 2001, 3307.
Brehm, I.; Hinneschiedt, S.; Meier, H. Eur. J. Org. Chem. 2002, 3162.
Forsén, S.; Merényi, F.; Nilsson, M. Acta Chem. Scand. 1964, 18, 1208.
Ng, S.; Lee, H.-H.; Bennett, G. J. Magn. Reson. Chem. 1990, 28, 337.
Ferreira, D.; Roux, D. G. J. Chem, Soc. Perkin Trans I 1977, 134.
Clemo, N. G.; Gedge, D. R.; Pattenden, G. J. Chem. Soc., Perkin Trans. 1 1981, 1448.
Li, X.-C.; ElSohly, H. N.; Nimrod, A. C.; Clark, A. M. J. Nat. Prod. 1999, 62, 767.
Marr, K. A., Lyons; C. N, Rustad, T; Bowden, R. A, White, T. C. Antimicrob. Agents Chemother. 1998, 42, 2584.
White T. C. Antimicrob. Agents Chemother. 1997, 41, 1482.
Pfaller, M. A.; Rhine-Chalberg, J.; Redding, S. W.; Smith, J.; Farinacci, G.; Fothergill, A. W.; Rinaldi, M. G. J. Clin. Micro. 1994, 32, 59.
Odds, F. C. Int. J. Std. AIDS 1992, 3, 157.
Coleman, D. C.; Bennett, D. E.; Sullivan, D. J.; Gallagher, P. J.; Henman, M. C.; Shanley, D. B.; Russell, R. J. Crit. Rev. Microbiol. 1993, 19, 61.
Nilsson, M. Acta Chem. Scand. 1964, 18:441.
Novikov, V. L.; Shestak, O. P.; Kamernitskii, A. V.; Elyakov, G. B. Izvestiya Akademii Nauk SSR, Seriya Khimicheskaya 1981, 1, 236.
Choi, Y. H.; Kwon, S. Y.; Kim, J. H.; Beak, N. I.; Choi, G. J.; Cho, K. Y.; Lee, B. M. Han'guk Nonghua Hakhoechi 2003, 46:151.
NCCLS, Reference Method for Broth Dilution Antifungal Susceptibility Testing of Yeasts; Approved Standard M27-A2. National Committee on Clinical Laboratory Standards, 2002 22 (15).
NCCLS, Reference method for broth dilution antifungal susceptibility testing of filamentous fungi; approved standard, M38-A. National Committee on Clinical Laboratory Standards, 2002, 22(16).
NCCLS, Methods for Dilution Antimicrobial Susceptibility Tests for Bacteria that Grow Aerobically M7-A5. National Committee on Clinical Laboratory Standards, 2000, 20(2).
NCCLS, Susceptibility Testing of Mycobacteria, Nocardia, and Other Aerobic Actinomycetes; Tentative Standard—Second Edition, M24-T2. National Committee on Clinical Laboratory Standards, 2000, 20(26).
Franzblau, S.G.; Witzig, Richard S.; Mclaughlin, James C.; Torres, Patricia; Madico, Guillermo; Hernandez, Antonio; Degnan, Michelle T.; Cook, Mary B.; Quenzer, Virginia K.; Ferguson, Robert M.; Gilman, Robert H. J. Clin. Microbiol.1998, 36, 362.

LandOfFree

Say what you really think

Search LandOfFree.com for the USA inventors and patents. Rate them and share your experience with other people.

Rating

Cyclopentenedione antifungal compounds and methods for their... does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Cyclopentenedione antifungal compounds and methods for their..., we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Cyclopentenedione antifungal compounds and methods for their... will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFUS-PAI-O-3573589

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.