Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Reexamination Certificate
2006-04-25
2006-04-25
Stockton, Laura L. (Department: 1626)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
C548S247000, C548S248000
Reexamination Certificate
active
07034046
ABSTRACT:
The present invention relates to compounds according to the general formula (I) which bind to the nuclear receptor, NR1H4, and act as agonists and antagonists of the NR1H4 receptor. The invention further relates to the treatment of diseases and/or conditions through binding of the nuclear receptor by the compounds.
REFERENCES:
patent: 4634783 (1987-01-01), Fujii et al.
patent: 5859257 (1999-01-01), Talley
patent: 6005103 (1999-12-01), Domagala et al.
patent: 6051574 (2000-04-01), Anthony
patent: 6201020 (2001-03-01), Zhang et al.
patent: 2002/0143020 (2002-10-01), Adams et al.
patent: 19943636 (2001-03-01), None
patent: 0098713 (1984-01-01), None
patent: 573883 (1993-12-01), None
patent: 11/263775 (1999-09-01), None
patent: WO-00/08001 (2000-02-01), None
patent: WO-00/37077 (2000-06-01), None
patent: WO-00/64876 (2000-11-01), None
CA Registry No. 433249-96-8, entry date into Registry file on STN is Jun. 22, 2002.
CA Registry No. 419538-90-2, entry date into Registry file on STN is May 21, 2002.
CA Registry No. 381677-00-5, entry date into Registry file on STN is Jan. 10, 2002.
CA Registry No. 354538-63-9, entry date into Registry file on STN is Sep. 4, 2001.
CA Registry No. 354538-61-7, entry date into Registry file on STN is Sep. 4, 2001.
CA Registry No. 348601-30-9, entry date into Registry file on STN is Jul. 26, 2001.
CA Registry No. 348602-52-8, entry date into Registry file on STN is Jul. 26, 2001.
CA Registry No. 339020-00-7, entry date into Registry file on STN is May 30, 2001.
CA Registry No. 338978-05-5, entry date into Registry file on STN is May 30, 2001.
CA Registry No. 324532-75-4, entry date into Registry file on STN is Feb. 27, 2001.
CA Registry No. 314027-56-0, entry date into Registry file on STN is Jan. 16, 2001.
CA Registry No. 314027-55-9, entry date into Registry file on STN is Jan. 16, 2001.
CA Registry No. 314027-54-8, entry date into Registry file on STN is Jan. 16, 2001.
CA Registry No. 313958-43-9, entry date into Registry file on STN is Jan. 15, 2001.
CA Registry No. 313958-42-8, entry date into Registry file on STN is Jan. 15, 2001.
CA Registry No. 312947-41-4, entry date into Registry file on STN is Jan. 5, 2001.
CA Registry No. 312947-40-3, entry date into Registry file on STN is Jan. 5, 2001.
CA Registry No. 312947-39-0, entry date into Registry file on STN is Jan. 5, 2001.
CA Registry No. 312947-38-9, entry date into Registry file on STN is Jan. 5, 2001.
CA Registry No. 312947-37-8, entry date into Registry file on STN is Jan. 5, 2001.
CA Registry No. 312947-36-7, entry date into Registry file on STN is Jan. 5, 2001.
CA Registry No. 302574-97-6, entry date into Registry file on STN is Nov. 13, 2000.
CA Registry No. 302573-71-3, entry date into Registry file on STN is Nov. 13, 2000.
CA Registry No. 261929-20-8, entry date into Registry file on STN is Apr. 14, 2000.
CA Registry No. 261929-19-5, entry date into Registry file on STN is Apr. 14, 2000.
CA Registry No. 219865-50-6, entry date into Registry file on STN is Feb. 21, 1999.
CA Registry No. 219499-05-5, entry date into Registry file on STN is Feb. 7, 1999.
CA Registry No. 219499-04-4, entry date into Registry file on STN is Feb. 7, 1999.
CA Registry No. 219499-03-3, entry date into Registry file on STN is Feb. 7, 1999.
CA Registry No. 219499-02-2, entry date into Registry file on STN is Feb. 7, 1999.
CA Registry No. 219499-01-1, entry date into Registry file on STN is Feb. 7, 1999.
CA Registry No. 219140-10-0, entry date into Registry file on STN is Feb. 5, 1999.
CA Registry No. 218928-39-3, entry date into Registry file on STN is Feb. 3, 1999.
CA Registry No. 216774-86-6, entry date into Registry file on STN is Jan. 10, 1999.
Lazzarini et al., CA 96:52213, 1982.
Pocar et al., CA 94:30610, 1981.
CA Registry No. 331974-09-5, entry date into Registry file on STN is Apr. 20, 2001.
CA Registry No. 94084-26-1, entry date into Registry file on STN is Jan. 5, 1985.
Roussel et al., CA 131:73522, 1999.
Yakhak Hoechi, “Analgesic, Anti-inflammatory and Antiviral Effects of Melandrin Derivatives”, Chemical Abstracts, vol. 121, No. 23, Dec. 5, 1994, (Columbus, OH, USA), p. 39, col. 1, the abstract No. 271343d.
Patrick R. Maloney et al., “Identification of a Chemical Tool for the Orphan Nuclear Receptor FXR”, Journal of Medicinal Chemistry, vol. 43, No. 16, Aug. 10, 2000, pp. 2971-2974, XP-002186187.
Bauer Ulrike
Cheruvallath Zach
Deuschle Ulrich
Dneprovskaia Elena
Gahman Tim
Phenex Pharmaceuticals AG
Saliwanchik Lloyd & Saliwanchik
Stockton Laura L.
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