Aminophenanthridinone and aminophenanthridine as NPY-5...

Details Aminophenanthridinone and aminophenanthridine as NPY-5... Aminophenanthridinone and aminophenanthridine as NPY-5...

2005-10-25

2005-10-25

Desai, Rita (Department: 1625)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

C546S108000, C546S110000

Reexamination Certificate

active

06958347

ABSTRACT:
The present invention provides NPY-5 receptor antagonists having a Formula (I)Methods and pharmaceutical compositions useful for treating diseases, conditions and/or disorders modulated by the above NPY-5 receptor antagonists are also provided.

REFERENCES:
patent: 5336674 (1994-08-01), Dininno et al.
patent: 5576337 (1996-11-01), Bruns, Jr. et al.
patent: 0759441 (1997-02-01), None
patent: 1033366 (2000-09-01), None
patent: 1184373 (2002-03-01), None
patent: WO 9901128 (1999-01-01), None
patent: WO 02096902 (2002-12-01), None
A. Balasubramaniam, Am. J. of Surgery, 183, pp. 430-434, 2002.
Flood and Morley Peptides, 10, pp. 963-966, 1989.
Leibowitz and Alexander, Peptides, 12, pp. 1251-1260, 1991.
Stanley et al., Peptides, 13, pp. 581-587, 1992.
McCauley and Westfal, J. Pharmacol, Exp. Ther. 261, pp. 863-868, 1992.
Grundemar et al., Br. J. Pharmacol, 105, pp. 45-50, 1992.
Grundemar and Hakanson, TIPS, May 1994, vol. 15, pp. 153-159.
Wahlestedt et al., Regul. Peptides, 13, pp. 307-318, 1986.
Redrobe et al., Life Sciences, 71, pp. 2921-2937, 2002.
M. Hammond et al, Bioorganic & Medicinal Chemistry Letters, 2003, vol. 13, pp 1989-1992, “Structure-Activity Relationships in a Series of NPY Y5 Antagonists: 3-Amido-9-ethylcarbazoles, Core-Modified Analogues and Amide Isosteres”.

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