Use of phenylheteroalkylamine derivatives

Details Use of phenylheteroalkylamine derivatives Use of phenylheteroalkylamine derivatives

Filed on

2005-10-11

Date issued

2005-10-11

Examiner

Richter, Johann (Department: 1626)

Patent Class

Drug, bio-affecting and body treating compositions

SubClass

Designated organic active ingredient containing

SubSubClass

Heterocyclic carbon compounds containing a hetero ring...

Other Related Categories

C514S374000, C514S524000, C514S649000, C548S235000, C544S167000, C558S418000, C558S422000

Type

Reexamination Certificate

Status

active

Patent number

06953797

Description

ABSTRACT:
There is disclosed the use of a compound of formula (I), wherein R1, R2, X, Y, V, W and Z are as defined in the specification, and pharmaceutically acceptable salts, enantiomers or racemates thereof, in the manufacture of a medicament, for the treatment or prophylaxis of diseases or conditions in which inhibition of nitric oxide synthase activity is beneficial. Certain novel compounds of formula (Ia) and pharmaceutically acceptable salts thereof, and enantiomers and racemates thereof are disclosed; together with processes for their preparation, compositions containing them and their use in therapy. The compounds of formulae (I) and (Ia) are inhibitors of the enzyme nitric oxide synthase and are thereby particularly useful in the treatment or prohylaxis of inflammatory disease

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