Melanin-concentrating hormone antagonist

Details Melanin-concentrating hormone antagonist Melanin-concentrating hormone antagonist

2005-08-16

2005-08-16

Seaman, D. Margaret (Department: 1625)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C546S162000, C546S163000, C546S169000, C514S311000, C514S312000, C514S313000

Reexamination Certificate

active

06930185

ABSTRACT:
A melanin-concentrating hormone antagonist comprising a compound of the formula (I):wherein Ar1is a cyclic group which may be substituted; X and Y are the same or different and are a spacer having a main chain of 1 to 6 atoms; Ar is a condensed polycyclic aromatic ring which may be substituted; R1and R2are the same or different and are hydrogen atom or a hydrocarbon group which may be substituted; or R1and R2, together with the adjacent nitrogen atom, may form a nitrogen-containing heterocyclic ring which may be substituted; or R2, together with the adjacent nitrogen atom and Y, may form a nitrogen-containing heterocyclic ring which may be substituted; or R2, together with the adjacent nitrogen atom, Y and Ar, may form a condensed ring; or a salt thereof is useful as an agent for preventing or treating obesity, etc.

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