Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1996-04-03
1998-01-27
Morris, Patricia L.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
514253, 514256, 514269, 514272, 514274, 544232, 544238, 544310, 544315, 544319, 544324, 544328, 544331, 544333, 544405, 546113, A61K 31435, C07D47104
Patent
active
057122857
ABSTRACT:
thereof by a methylene group to a tetrahydropyridinyl moiety, the latter moiety being substituted in turn by an aryl- or heteroaryl-substituted divalent monocyclic radical, are ligands for dopamine receptorsubtypes within the body, in particular the D.sub.4 subtype, and are accordingly of use in the treatment and/or prevention of disorders of the dopamine system, including schizophrenia and depression.
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Curtis Neil Roy
Kulagowski Janusz Jozef
Leeson Paul David
Ridgill Mark Peter
Merck Sharp & Dohme Ltd.
Morris Patricia L.
North Robert J.
Winokur Melvin
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