Benzothiopene compounds, compositions, and method of inhibiting

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

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514212, 5142388, 514422, 514443, 560609, 544146, 546202, 548525, 548527, 549 51, 549 58, A61K 31445, A61K 3140, C07D40912

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active

054847982

ABSTRACT:
The present invention provides novel benzothiophene compounds of formula I ##STR1## wherein R is --H, --OH, --O(C.sub.1 -C.sub.4 alkyl), --O--CO--(C.sub.1 -C.sub.6 alkyl), --O--CO--Ar in which Ar is optionally substituted phenyl, or --O--SO.sub.2 --(C.sub.4 -C.sub.6 alkyl);

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