Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1995-02-06
1997-09-02
Rotman, Alan L.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
546 70, C07D47104, A61K 3144
Patent
active
056631782
ABSTRACT:
The present invention provides novel tetrahydro-beta-carboline compounds having useful central nervous system activity. Further, there is provided tetrahydro-beta-carboline related compounds which are useful intermediates and have beneficial central nervous system activity. The invention provides formulations and methods for using the novel tetrahydro-beta-carboline and related compounds. Such compounds are particularly useful for the modulation of a 5-HT.sub.2B receptor.
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Derwent Abstract 84-115276/19 Oct. 29, 1982 DE-3240-514-A.
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Audia James E.
Baker Stephen Richard
Carrera Jesus Ezquerra
Pedregal Tercero Concepcion
Peteira Carlos Lamas
Boone David E.
Eli Lilly and Company
Rotman Alan L.
Vorndran-Jones MaCharri
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