Preparation of 2-halo-5-methylpyridines from 4-methyl-4-pentene

Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...

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560130, 560184, 560226, C07D30340

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active

047090634

ABSTRACT:
A method of preparing certain 2-halo-5-methylpyridines, useful as herbicide intermediates, is presented starting from acyclic pentenes. The pentene is difunctionalized, e.g., by making the epoxide, and is then reacted with a nitrogen source to close the ring. The nitrogen-containing 6-membered heterocycle may then be aromatized readily to produce the 2-halo-5-methylpyridine desired. Also part of the invention are novel acyclic and cyclic intermediates used in the process.

REFERENCES:
patent: 3642833 (1972-02-01), Wuiff et al.
patent: 4234741 (1980-11-01), Petrzilka
John J. Ritter et al., Jour. Org. Chem., vol. 27, Feb. 1962, pp. 622-623.
M. Julia et al., Bulletin de la Societe Chimique de France (1969), No. 7, pp. 2415-2427.
W. S. Johnson et al., Jour. Am. Chem. Soc., vol. 92 (1970), pp. 741-743.
J. E. McMurry et al., J. Org. Chem., vol. 40(17), (1975), pp. 2556-2557.
Isagulyants, V. I. et al., Dok. Akad. Nauk Arm., vol. 44, 1967, pp. 115-120.
Kuehne, Martin E. et al., J. Org. Chem., vol. 45, 1980, pp. 3259-3265.

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