Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1996-02-21
1997-07-08
Haley, Jacqueline
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
548427, 548430, C07D20958, A61K 3140
Patent
active
056461739
ABSTRACT:
The invention relates to tricyclic pyrrole derivatives useful as 5-HT selective agents of the formula ##STR1## wherein R.sup.1 to R.sup.4 are, independently, hydrogen, halogen, lower alkyl, phenyl, cycloalkyl or lower alkoxy and R.sup.2 additionally is lower alkoxycarbonyl, acyloxy or mesyloxy;
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Bos Michael
Wichmann Jurgen
Widmer Ulrich
Ciambrone Coletti Ellen
Haley Jacqueline
Hoffmann-La Roche Inc.
Johnston George W.
Silverman Robert A.
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