Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1995-05-26
1997-04-08
Gupta, Yogendra N.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
5462774, 546266, 5462714, 5462721, 5462724, 5462727, 5462754, 546113, 5462804, 546152, 5462684, 5462717, 5462677, 5462687, 5462691, 5462701, 546314, 5462814, 546339, 5462697, 5462711, 5462834, 514256, 514269, 514300, 514311, 514314, 514338, 514340, 514354, 514406, 514415, 544242, 544333, 544335, 5483731, 548509, A61K 3144, A61K 31505, C07D21316, C07D23926
Patent
active
056188218
ABSTRACT:
Compounds of the formula ##STR1## wherein Q is chosen from the group consisting of pyridyl, pyrazyl, pyrimidyl, quinolyl, indolyl and 7-azaindolyl or any of these substituted with one or two substituents;
Y is an alkylene bridge of 3-9 carbon atoms;
R.sub.1 and R.sub.2 are each independently chosen from hydrogen, halo, alkyl, alkenyl, amino, alkylthio, hydroxy, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl, alkylsulfinylalkyl, alkylsulfonylalkyl, alkoxy, nitro, carboxy, alkoxycarbonyl, dialkylaminoalkyl, alkylaminoalkyl, aminoalkyl, difluoromethyl, trifluoromethyl or cyano;
R.sub.3 is alkoxycarbonyl, alkyltetrazolyl, substituted or unsubstituted phenyl or heterocyclyl, the N-oxide thereof, or a pharmaceutically acceptable acid addition salt thereof is an effective antipicornaviral agent.
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Aldous David J.
Bailey Thomas R.
Diana Guy D.
Kuo Gee-Hong
Nitz Theodore J.
Davis William J.
DuPont Paul E.
Gupta Yogendra N.
Sanofi (S.A.)
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