Chiral, N-protected, N-substituted .alpha.-amino acids

Details Chiral, N-protected, N-substituted .alpha.-amino acids Chiral, N-protected, N-substituted .alpha.-amino acids

1983-05-23

1985-08-13

Shippen, Michael L.

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

548477, 548497, 260465D, 2604654, 260464, 560 16, 560 24, 560 29, 560 32, 560 33, 560 45, 560148, 560158, 560159, 560160, 560163, 560165, 562426, 562439, 562444, 562450, 562507, 562557, 562560, 562561, 562567, 562571, 562574, C07C125065, C07C10346

Patent

active

045351678

ABSTRACT:
Chiral N-protected, N-substituted .alpha.-amino acids are described. These compounds are prepared by condensation of an N-protected .alpha.-amino acid with an aldehyde followed by the selective reductive cleavage of an oxazolidinone intermediate.

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