Preparation of metallated and substituted alkynes

Organic compounds -- part of the class 532-570 series – Organic compounds – Silicon containing

Patent

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

568687, 585505, C07F 704, C07C 4100

Patent

active

051625628

ABSTRACT:
A process is provided for making metallated and substituted alkynes from feedstocks which include alkadienes containing allenic unsaturation or such alkadienes in a mixture with alkynes having either internal or terminal unsaturation, such as a mixture of propadiene and propyne. This reaction involves an initial step in which the allenic hydrocarbon and any internal alkyne is isomerized and simultaneously the resultant terminal alkynes are metallated with an alkali metal. The reaction is carried out at relatively low temperatures in a suitable inert solvent such as diethylether. When metallation is complete the reaction mixture can be contacted directly with any suitable electrophile, such as a halo silane, for example, chlorotrimethylsilane, and the alkali metal on the terminal alkyne is replaced with the desired substituent. The products thus formed are useful as monomers for preparing polymers having a variety of properties, for example, as asymmetric membranes for gas separation.

REFERENCES:
patent: 3410918 (1968-11-01), Beumel, Jr. et al.
patent: 3671605 (1972-06-01), Smith, Jr.
patent: 3752848 (1973-08-01), Smith, Jr.
patent: 4036904 (1977-07-01), Strope
patent: 5062998 (1991-11-01), Herman et al.
Collignon et al., Bull. Soc. Chim. Fr., (1-2, Pt. 2) pp. 120-124 [See FIG. #3 p. 121].
Fitzmaurice et al., J. Organometal, Chem. 285 (1985) 375-381.
Rajagopalan et al. Synthesis, (1984) 111.
Z. L. Deph et al., "In Spectra of Catalysts and Corabid Molecule 25. Isomerization of Allene and Methylacetylene Aluminum Oxide", Izo. Akad. Nauk. 555 R, Lir. Khim (1978) 111, 24073.
C. P. Khulbe, et al., "Allene-methylacetylene isomerization over silica-supported cobalt and iron catalysts", /Canadian Journal of Chemistry, vol. 56, No. 22, Nov. 15, 1978, p. 2791.
C. A. Brown, et al., "The Acetylene Zipper, An Excetpionally Facile Contrathermodynamic Multipositional Isomerization of Alkynes with Potassium 3-Aminopropylamide", J. Am. Chem. Soc. p. 891, (1975) 97.
S. R. Macaulay, "The rearrangement of isomeric linear decyn-1-ols by reaction with the sodium salt of 1,3-diaminopropane;" Can. of Chem., 1980 National Research Council of Canada, p. 2567, 58.
S. R. Abrams, "Alkyne isomerization reagents: alkal metal amides", Can. J. Chem., vol. 62, p. 1333, (1984).
S. R. Abrams, "Isomerization of actylenic acids with sodium salt of 1,2-diaminoethane: a one step synthesis of megatomoic acid," Can. J. Chem., p. 1238, (1984) 62.
J. H. Wotiz, "The Mechanism of the Base-Catalyzed Prototropic Propargylic Rearrangement in Vicinal Diamines", J. Org. Chem., vol. 38, No. 3, 1973, p. 489.
S. R. Abrams et al., "On the Mechanism of 1,3-Prototropic Shifts in Acetylene-Allene Isomerizations", J. Org. Chem., 1987, 52, p. 1835.

LandOfFree

Say what you really think

Search LandOfFree.com for the USA inventors and patents. Rate them and share your experience with other people.

Rating

Preparation of metallated and substituted alkynes does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Preparation of metallated and substituted alkynes, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Preparation of metallated and substituted alkynes will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFUS-PAI-O-2295219

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.