Substituted 1-phenyl-3-pyrazolecarboxamides active on neurotensi

Details Substituted 1-phenyl-3-pyrazolecarboxamides active on neurotensi Substituted 1-phenyl-3-pyrazolecarboxamides active on neurotensi

Filed on

1996-04-10

Date issued

1998-03-03

Examiner

Richter, Johann

Patent Class

Drug, bio-affecting and body treating compositions

SubClass

Designated organic active ingredient containing

SubSubClass

Having -c-, wherein x is chalcogen, bonded directly to...

Other Related Categories

5483731, 5483751, 5483761, 5483771, A61K 31415, A01N 4356, C07D23114

Type

Patent

Status

active

Patent number

057234833

Description

ABSTRACT:
The invention relates to new substituted 1-phenyl-3-pyrazolecarboxamides having a great affinity for human neurotensin receptors, to a process for preparing them and to pharmaceutical compositions containing them as active principles. More particularly, this invention relates to the discovery that the affinity for neurotensin receptors, especially human neurotensin receptors, is increased by substituting the phenyl group of 1-phenyl-3-pyrazolecarboxamide compounds with particular groups.

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