Process for the preparation of imidazobenzodiazepines

Details Process for the preparation of imidazobenzodiazepines Process for the preparation of imidazobenzodiazepines

1980-02-21

1981-03-31

Rollins, Alton D.

Chemistry of carbon compounds

Miscellaneous organic carbon compounds

C-metal

2602456, 2602457, C07D48704

Patent

active

042592410

ABSTRACT:
A multistep process is presented for the preparation of imidazobenzodiazepines of the formula ##STR1## wherein X is selected from the group consisting of hydrogen, halogen, nitro and trifluoromethyl; Y is selected from the group consisting of hydrogen, halogen or trifluoromethyl; R.sub.1 is hydrogen or lower alkyl and R.sub.2 is a disubstituted amine.
Also presented are novel intermediates utilized in the process.
The end products and intermediates are useful as sedatives, anxiolytics, muscle relaxants and anticonvulsants.
The end products are especially useful in intravenous compositions for use in preoperative anesthesia.

REFERENCES:
patent: 4125726 (1978-11-01), Walser

Affiliated with

Also associated with

Rating

Process for the preparation of imidazobenzodiazepines does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Process for the preparation of imidazobenzodiazepines, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Process for the preparation of imidazobenzodiazepines will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-2242333