Benzothiazepine derivatives

Details Benzothiazepine derivatives Benzothiazepine derivatives

1992-10-14

1995-01-03

Shah, Mukund J.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

540491, A61K 3155, C07D41706

Patent

active

053786980

ABSTRACT:
A compound of the formula: ##STR1## wherein X is .dbd.N--A--R.sup.1 or .dbd.C(R.sup.1)R.sup.2 ; A is a single bond, polymethylene or --CO--; R.sup.1 and R.sup.2 are each hydrogen, C.sub.1 -C.sub.6 alkyl, C.sub.3 -C.sub.7 cycloalkyl, unsubstituted or substituted phenyl, optionally substituted benzhydryl, or optionally substituted 5 to 6 membered heterocyclic group; Y is hydrogen, halogen, C.sub.1 -C.sub.6 alkyl, C.sub.3 -C.sub.7 cycloalkyl, C.sub.1 -C.sub.6 alkoxy, optionally substituted phenoxy, optionally substituted benzyloxy, or optionally substituted benzyl; Z is hydrogen or acyl; n is an integer of from 2 to 6, and pharmaceutically acceptable salt thereof. A pharmaceutical composition containing the compound, which is useful for treating hypertension and cardiac diseases, is also provided.

REFERENCES:
patent: 4567175 (1986-01-01), Takeda et al.
patent: 4584131 (1986-04-01), Floyd et al.
patent: 4594342 (1986-06-01), Takeda et al.
patent: 4963545 (1990-10-01), Zobrist et al.
patent: 5001236 (1991-03-01), Borcherding et al.
patent: 5063225 (1991-11-01), Clemence

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