Tricyclic vasopressin agonists

Details Tricyclic vasopressin agonists Tricyclic vasopressin agonists

1998-07-24

2000-07-18

Shah, Mukund J.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

514 63, 540548, A61K 31553, C07D49802, A61P 710

Patent

active

060908033

ABSTRACT:
The present invention provides compounds of the general formula: ##STR1## wherein W is O or NH, optionally substituted, as well as methods and pharmaceutical compositions utilizing these compounds for the treatment of disorder which may be remedied or alleviated by vasopressin agonist activity, including diabetes insipidus, nocturnal enuresis, nocturia, urinary incontinence, bleeding and coagulation disorders, or temporary delay of urination.

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