Triazolo quinoxalines and their preparation and use

Details Triazolo quinoxalines and their preparation and use Triazolo quinoxalines and their preparation and use

1994-08-03

1996-04-02

Berch, Mark L.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

544346, 544354, A61K 31495, C07D48704, C07D24152

Patent

active

055040853

ABSTRACT:
Quinoxaline compounds represented by formulas I or II, ##STR1## wherein R.sup.1 and R.sup.2 are independently hydrogen, C.sub.1-6 -alkyl, halogen, NO.sub.2, NH.sub.2, CN, CF.sub.3, SO.sub.2 NR.sup.4 R.sup.5 wherein R.sup.4 and R.sup.5 are independently hydrogen or C.sub.1-6 -alkyl, or COR.sup.6 wherein R.sup.6 is C.sub.1-6 -alkyl; and R.sup.3 is hydrogen, C.sub.1-6 -alkyl or CF.sub.3, compositions thereof and methods of preparing the compounds are described.
The compounds are useful in the treatment of indications caused by hyperactivity of the excitatory neurotransmitters.

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