Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Patent
1989-01-17
1991-01-01
Daus, Donald G.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
5142292, 544 34, 544 48, 544101, 544105, C07D51304
Patent
active
049818503
ABSTRACT:
Substituted 1,2,4-triazolo[1,5-c]pyrimido[1,4]-azines have been found to have potent bronchodilator activity. Also, pharmacological methods for inducing bronchodilation using such compounds, pharmaceutical compositions containing such compounds, and synthetic intermediates, including 1,2,4-triazolo[4,3-c]-pyrimido[1,4]azines, for preparing such compounds.
REFERENCES:
patent: 4276292 (1981-06-01), St. Georgieu
patent: 4477450 (1984-10-01), Wade
patent: 4503050 (1985-03-01), Wade
patent: 4547499 (1985-10-01), Hester
patent: 4572910 (1986-02-01), Wade
patent: 4639445 (1987-01-01), McQuinn
patent: 4734413 (1988-03-01), Wade
Chem. Abstr, vol. 94, entry 1922806 (1981).
Sazonov et al., Khimiya Geterotsiklicheskikh, 1973, 171.
Sazonov et al., Khimiya Geterotsiklicheskikh, 1972, 1285.
Sazonov et al., Khimiya Geterotsiklicheskikh, 1976, 681.
Melik-Ogandzhanyan et al., Khimiya Geterotsiklicheskikh Soedinenii, 1985, 974.
E. F. Schroeder and R. M. Dodson, J. Amer. Chem. Soc., 84, 1904-1913 (1962).
R. N. Henri, R. A. Lazarus and S. J. Benkovic, J. Med. Chem., 26, 559-563 (1983).
Daus Donald G.
Kirn Walter N.
Riker Laboratories Inc.
Sell Donald M.
Sprague Robert W.
LandOfFree
Triazolo[1,5-c]pyrimido[1,4]azines as bronchodilators does not yet have a rating. At this time, there are no reviews or comments for this patent.
If you have personal experience with Triazolo[1,5-c]pyrimido[1,4]azines as bronchodilators, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Triazolo[1,5-c]pyrimido[1,4]azines as bronchodilators will most certainly appreciate the feedback.
Profile ID: LFUS-PAI-O-1996413