Substituted 3-(aminoalkylamino)-1,2-benzisoxazoles and related c

Details Substituted 3-(aminoalkylamino)-1,2-benzisoxazoles and related c Substituted 3-(aminoalkylamino)-1,2-benzisoxazoles and related c

1997-06-19

1998-05-26

Grumbling, Matthew V.

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

544283, C07D26120

Patent

active

057567549

ABSTRACT:
This application relates to compounds of the formula ##STR1## wherein R.sup.1, X, Y and n are as defined in the specification; and pharmaceutically acceptable addition salts thereof and optical and geometric isomers or racemic mixtures thereof; which compounds are useful for the treatment of various memory dysfunctions characterized by a decreased cholinergic function such as Alzheimer's disease. Compounds of this invention also inhibit monoamine oxidase and hence are useful as antidepressants.

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