Prodrugs of 3,4-hydroxy benzoyloxypropanolamines

Details Prodrugs of 3,4-hydroxy benzoyloxypropanolamines Prodrugs of 3,4-hydroxy benzoyloxypropanolamines

1988-12-15

1990-01-30

Daus, Donald G.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

5142378, 514330, 514374, 514451, 514452, 514428, 514487, 544162, 546237, 548215, 548237, 548538, 549372, 549425, 549487, 560110, A61K 3124, C07C10148

Patent

active

048974170

ABSTRACT:
In accordance with the present invention, disclosed herein are compounds of the formula ##STR1## wherein R is straight or branched loweralkyl, R.sub.1 is hydrogen, straight or branched loweralkyl, lowercycloalkyl, amino, loweralkoxy or acylamino, and R.sub.2 is straight or branched loweralkyl, amino, cyclohexyl, morpholino, piperidino, tetrahydrofuranyl, dihydrofuranyl, tetrahydropyranyl, dioxolanyl, 2,2-dimethyl dioxolanyl, dioxanyl, pyrrolidinyl, tetrahydrooxazolyl, and dihydrooxazolyl, and pharmaceutically acceptable salts thereof. The compounds are useful in the treatment of glaucoma.

REFERENCES:
patent: 4195085 (1980-03-01), Stone
patent: 4402974 (1983-09-01), Matier et al.
patent: 4405642 (1983-09-01), Kam et al.
patent: 4579867 (1986-01-01), Escobar
patent: 4582855 (1986-04-01), Kam et al.
patent: 4661513 (1987-04-01), Berthold

Affiliated with

Also associated with

Rating

Prodrugs of 3,4-hydroxy benzoyloxypropanolamines does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Prodrugs of 3,4-hydroxy benzoyloxypropanolamines, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Prodrugs of 3,4-hydroxy benzoyloxypropanolamines will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-1923768