Tricyclic amide and urea compounds useful for inhibition of G-pr

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

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5142282, 514253, 5142328, 514256, 514274, 546 93, 544 586, 544361, 544126, 544405, 544333, 544316, 544238, C07D40114, C07D40106, A61K 31445

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057008060

ABSTRACT:
Novel compounds of Formula (7.0a), (7.0b) or (7.0c): ##STR1## are disclosed. Also disclosed is a method of inhibiting Ras function and therefore inhibiting the abnormal growth of cells. The method comprises administering a compound of the formula (7.0a), (7.0b) or (7.0c) to a biological system. In particular, the method inhibits the abnormal growth of cells in a mammal such as a human being.

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