Stereospecific synthesis of carboxyalkyl peptides

Details Stereospecific synthesis of carboxyalkyl peptides Stereospecific synthesis of carboxyalkyl peptides

1986-12-19

1989-01-31

Phillips, Delbert R.

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

548532, 548533, 548534, 558232, 558242, 560 33, 560 38, 560 41, 560165, 560169, 564152, 564153, 564154, 564157, 564159, C07D20954, C07D20700, C07C12506, C07C10102, C07C10126, C07C10319, C07C10300, C07C10320, C07C10307

Patent

active

048017213

ABSTRACT:
Methods for the alkylation of substituted amines with trifluorate esters is disclosed.

REFERENCES:
patent: 3419595 (1968-12-01), Hansen
patent: 3803199 (1974-04-01), Voss et al.
patent: 3810939 (1974-05-01), Ray-Chaudlin
patent: 3853939 (1974-12-01), Partos
patent: 4125555 (1978-11-01), Reineke
patent: 4310461 (1982-01-01), Krapcho et al.
patent: 4374829 (1983-09-01), Harris et al.
patent: 4390695 (1983-06-01), Krapcho et al.
patent: 4410520 (1983-10-01), Watthey
patent: 4415496 (1983-11-01), Harris et al.
patent: 4428940 (1984-01-01), Markwell
patent: 4431644 (1984-02-01), Smith et al.
patent: 4431645 (1984-02-01), Smith et al.
patent: 4440759 (1984-04-01), Omura et al.
patent: 4512924 (1985-04-01), Attwood et al.
Effenberger, V. et al., "Trifluoromethanesulfonate von -Hydroxy-Carbon Sauereestern" Agnew Chem., 95:50 (1983).
Howells, R. D. et al., "Trifluoromethanesulfonic Acid and Derivatives," Chem. Revs. 77(1):69 (1977).
Hansen, R. "Perfluoroalkanesulfonate Esters as Alkylating Agents", J. Org. Chem. 30:4322 (1965).
Burdon, J. et al., "Trifluoromethanesulfonate Esters and Their Alkylating Properties", Tetrahedron 21:1 (1965).
Kato, T. et al., Tetrahedron Letters 48:4741 (1978).
Schroder et al., The Peptides, vol. 1 (Academic Press), p. 181 (1965).
Merrifield, R. B., Advanced Enzymology "Solid Phase Peptide Synthesis", 32:221 (1969).
"Methoden der Organischen Chemie" (Houben-Weyl) vol. XV, part 1, p. 376 (1974).
Ohzeki, M. et al. "Stereochemical Studies", Chem. Pharm. Bull. 25(10):2676 (1977).
Fontana, A., "Selective Removal of Sulphur Protecting Groups of Cysteine Residues by Sulphenyl Halides", J.C.S. Chem. Comm. 976 (1975).
Urbach, H. et al., Tetrahedron Letters 25 (11):1143 (1984).
Hovius, K. et al., "Facile Intermolecular at .alpha.-Sulfonyl Carbon", Tetrahedron Letters 24:2477 (1972).
Beard, C. et al., "Synthesis of Some Novel Trifluoromethanesulfonates", J. Org. Chem. 38(21):3673 (1973).
Baldwin, J. et al., "Use of (S)-(Trifloxymethyloxirane in Synthesis", J. Med. Chem. 25(8):931 (1982).
Shiori, T. et al., "Diphenylphosphoxyl Azide", J. Amer. Chem. Soc. 94 (17):6203 (1972).
Katsuhara, Y. et al. "Stereochemistry of the Reaction of Chlorine(I) Trifluoromethanesulfonate", J. Am. Chem. Soc. 101(4):1039 (1979).

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