Pyrazolo(3,4-d)pyrimidine compounds, compositions and method of

Details Pyrazolo(3,4-d)pyrimidine compounds, compositions and method of Pyrazolo(3,4-d)pyrimidine compounds, compositions and method of

1988-04-14

1990-02-27

Shah, Mukund J.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

544262, C07D48704, A61K 31505

Patent

active

049046667

ABSTRACT:
The present invention provides pyrazolo[3,4-d]-pyrimidines of the general formula: ##STR1## wherein R.sub.1 is a C.sub.1 to C.sub.6 -alkyl radical, a C.sub.2 to C.sub.6 -alkenyl radical, a C.sub.3 to C.sub.7 -cycloalkyl radical or an aryl radical, R.sub.2 is a C.sub.2 to C.sub.6 -alkenyl radical, a C.sub.3 to C.sub.7 -cycloalkyl radical or an aralkyl or hetaralkyl radical with 1 to 6 carbon atoms in the alkyl moiety and substituted, if desired, one or more times by halogen, C.sub.1 to C.sub.6 -alkyl, hydroxyl, C.sub.1 to C.sub.6 -alkoxy, C.sub.1 to C.sub.3 -haloalkyl, C.sub.3 to C.sub.7 -alkoxy carbonyl, aminocarbonyl, C.sub.2 to C.sub.7 -alkylaminocarbonyl, C.sub.3 to C.sub.13 -dialkylaminocarbonyl, cyano or C.sub.1 to C.sub.6 -alkylthio and R.sub.3 is a hydrogen atom or a C.sub.2 to C.sub.6 -alkyl radical substituted, if desired, one or more times by hydroxyl or is a tetrahydrofuranyl or tetrahydropyranyl radical, with the proviso that R.sub.2 cannot be an unsubstituted benzyl radical when R.sub.1 is a methyl radical, and the physiologically acceptable salts thereof with inorganic and organic acids.
The present invention also provides processes for the preparation of these compounds and pharmaceutical compositions containing them.

REFERENCES:
patent: 3682918 (1972-08-01), Druey et al.
patent: 3720674 (1973-03-01), Breuer et al.

Affiliated with

Also associated with

Rating

Pyrazolo(3,4-d)pyrimidine compounds, compositions and method of does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Pyrazolo(3,4-d)pyrimidine compounds, compositions and method of , we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Pyrazolo(3,4-d)pyrimidine compounds, compositions and method of will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-174406