Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1992-06-16
1993-07-06
Tsang, Cecilia
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
514253, 544295, 544368, 548207, 548209, 548241, A61K 31495, A61K 31505, C07D40304, C07D27504
Patent
active
052254127
ABSTRACT:
Novel benzisothiazole- and benzisoxazole-3-carboxamides, processes and intermediates for the preparation thereof, and methods of treating psychoses utilizing compounds and compositions thereof are disclosed.
REFERENCES:
patent: 2626260 (1953-01-01), Clinton
patent: 3145215 (1964-08-01), Kirchner
patent: 3576810 (1971-04-01), Duncan
patent: 4021552 (1977-05-01), Welstead
patent: 4327103 (1982-04-01), Helsley
patent: 4452799 (1984-06-01), Temple
patent: 4710500 (1987-12-01), Perregaard
patent: 4758503 (1988-07-01), Sato
patent: 4954503 (1990-09-01), Strupczewski et al.
patent: 5008264 (1991-04-01), Davis
patent: 5030639 (1991-07-01), Davis
patent: 5077405 (1991-12-01), Strupczewski et al.
patent: 5114936 (1992-05-01), Wettlaufer et al.
patent: 5130315 (1992-07-01), Ong et al.
U.S. patent application Ser. No. 639,639 filed by H. H. Ong, et al., Jan. 10, 1991.
L. Amoretti, et al., Il Farmaco (Ed. Sc.), vol. 27, pp. 855 to 869, published Oct., 1972, entitled, "Biological Properties of 1,2-Benzisothiazole Compounds," and English translation.
E. Molina, et al., Acta Bio-Med., vol. 45, pp. 183 to 191, published 1974, entitled, "Biological Properties of 1,2-Benzisothiazole Compounds. Spasmolytic Activity of Benzisothiazol-3-carboxamides," and English translation.
J. P. Yevich, et al., Journal of Medicinal Chemistry, vol. 29, pp. 359 to 369, published 1986, entitled "Synthesis and Biological Evaluation of 1-(1,2-Benzisothiazol-3-yl) and (1,2-Benzisoxazol-3-yl)piperazine Derivatives as Potential Antipsychotic Agents".
J. T. Strupczewski, et al., Journal of Medicinal Chemistry, vol. 28, pp. 761 to 769, published 1985, entitled, "Synthesis and Neuroleptic Activity of 3-(1-Substituted-4-piperidinyl)-1,2-benzisoxazoles".
Hrib Nicholas J.
Jurcak John G.
Hoechst-Roussel Pharmaceuticals Incorporated
Tsang Cecilia
Wittekind Raymond R.
LandOfFree
Benzoisothiazole-and benzisoxazole-3-carboxamides does not yet have a rating. At this time, there are no reviews or comments for this patent.
If you have personal experience with Benzoisothiazole-and benzisoxazole-3-carboxamides, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Benzoisothiazole-and benzisoxazole-3-carboxamides will most certainly appreciate the feedback.
Profile ID: LFUS-PAI-O-1689710