Process for the production of chiral hydroxy-.beta.-lactams and

Details Process for the production of chiral hydroxy-.beta.-lactams and Process for the production of chiral hydroxy-.beta.-lactams and

1992-02-27

1994-03-15

Dees, Jose G.

Organic compounds -- part of the class 532-570 series

Organic compounds

Carboxylic acids and salts thereof

C07C22900

Patent

active

052947378

ABSTRACT:
The reaction between a hydroxyacetic acid derivative bearing an oxygen protecting group and a chiral auxiliary group and an imine produces chiral .beta.-lactams. Hydrolysis of the chiral .beta.-lactams produces chiral amino acid analogs.

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