Process for optically active 2-alkyl-2,5-diazabicyclo[2.2.1]hept

Details Process for optically active 2-alkyl-2,5-diazabicyclo[2.2.1]hept Process for optically active 2-alkyl-2,5-diazabicyclo[2.2.1]hept

1994-09-06

1995-12-12

Springer, David B.

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C07D48708

Patent

active

054751179

ABSTRACT:
1S,4S and 1R,4R-2-Alkyl-2,5-diazabicyclo[2.2.1]heptanes useful as intermediates in the synthesis of certain antibacterial quinolones, are prepared respectively, from trans-4-hydroxy-L-proline and trans-4-hydroxy-D-proline via multistep procedures.

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