Process for preparing quinoline amines

Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...

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546155, 546157, 546159, C07D47104, C07D21520, C07D21536, C07D21538

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active

053959370

ABSTRACT:
A process that involves reacting a 3-nitroquinoline-2,4-disulfonate with an amine or a substituted amine to selectively aminate at the 4-position to yield 1H-imidazo[4,5-c]quinolin-4-amines is disclosed.

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