Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1992-02-24
1993-05-04
Robinson, Allen J.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
549 52, 549 53, 549 54, 549 55, 549 56, A61K 3138, C07D33356
Patent
active
052082539
ABSTRACT:
3-Alkyloxy-, aryloxy-, or arylalkyloxy-benzo[b]thiophene-2-carboxamides are described as agents which block leukocyte adherence to vascular endothelium and, as such, are effective therapeutic agents for treating inflammatory diseases. Certain of these compounds are novel and methods of preparation are also described.
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Boschelli Diane H.
Connor David T.
Wright Clifford D.
Daignault Ronald A.
Robinson Allen J.
Russell Mark W.
Warner-Lambert & Company
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